- 英文名称
- Tibolone
- 分子式
- C21H28O2
- 分子量
- 312.45
- 中文别名
- 甲异炔诺龙; 甲基异炔诺酮; 甲基异炔酮; 17-羟基-7alpha-甲基-19-去甲孕甾-5(10)-烯-20-炔-3-酮; 提伯龙; 17-Hydroxy-7α-methyl-19-nor-17α-pregn-5(10)-en-20-yn-3-one; 7a-Methyl-5,10-norethindrone; 7a-Methyl-17a-ethynyl-17b-hydroxy-19-norandrost-5(10)-en-3-one; LIVIELLA; Org OD 14; (7α,17α)-17-Hydroxy-7-methyl-19-norpregn-5(10)-en-20-yn-3-one; 7a-Methyl-D5,10-norethindrone; (7R,8R,9S,13S,14S,17R)-17-Ethynyl-17-hydroxy-7,13-dimethyl-1,2,4,6,7,8,9,11,12,13,14,15,16,17-tetradecahydro-3H-cyclopenta[a]phenanthren-3-one; Livial; 7a-Methyl-17a-ethynyl-17b-hydroxyestr-5(10)-en-3-one; 5(10)-ESTREN-7-ALPHA-METHYL-17-ALPHA-ETHYNYL-17-BETA-OL-3-ONE; (7A,17A)-17-HYDROXY-7-METHYL-19-NORPREGN-5(10)-EN-20-YL-3-ONE; 17ALPHA-HYDROXY-7ALPHA-METHYL-19-NORPREGN-5(10)-EN-20-YN-3-ONE; 19-NORPREGN-5(10)-EN-20-YN-3-ONE,17-HYDROXY-7-METHYL-, (7A,17A)-
- 用途
- 生命科学;医药,雄激素、同化激素类药,用于治疗妇女更年期综合症,还能预防骨质疏松;用于子宫肌瘤(肌瘤<3cm患者可使用并定期监测,>4cm者需权衡利弊短期使用);用于子宫内膜异位症(缓解盆腔疼痛);用于下丘脑促性腺激素释放激素的反向添加(缓解绝经症状、预防骨质疏松)