4-碘-2-硝基苯胺为胺类衍生物，可用作有机试剂。
有机试剂
合成路线 1（1. 合成：20691-72-9）
产率：98%
合成条件：With sodium periodate; sulfuric acid; iodine; potassium iodide; sodium sulfite In water; acetic acid at 25℃; for 4 h;
实验步骤：一般步骤：在Na 2 SO 3存在下对苯酚（1d）进行碘化（典型程序）。 向100mL圆底烧瓶中加入3mmol苯酚在10mL乙酸中的溶液，以及KI3和Na2SO3溶液（预先通过向溶液中加入3mmol碘和3mmol Na2SO3制备） 迅速加入3毫升碘化钾在3毫升水中的溶液。 同时，加入3mmol NaIO4在5mL水中的溶液，并使用压力平衡滴液漏斗快速加入0.5mL硫酸。 将混合物在25℃下搅拌，通过TLC监测反应进程。 当反应完成时，将混合物倒入冰冷的水中，通过真空过滤分离固体产物，用去离子水洗涤两次，并干燥。
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