N-苯乙基氨基甲酸乙酯主要用于医药相关研究，作为有机合成中间体或药物分子前体，在多种药物研发项目中发挥作用（如通过酰化反应构建特定药效基团）。
医药研究
合成路线 1（1. 合成：6970-83-8）
产率：96%
合成条件：With triethylamine In dichloromethane at 0 - 20℃;
实验步骤：化合物2a-2h，3a-3h，4a-4h，5a-5h，6a-6h，7a-7h，11a-h和12a-12h的通用方法。 将10mL二氯甲烷和搅拌棒加入100-200mg胺中。 然后加入2当量的三乙胺，并在搅拌下将反应混合物冷却至0℃。 然后，将0.9当量的氯甲酸酯，异氰酸酯或硫代异氰酸酯滴加到反应混合物中，并使其缓慢升温至室温并继续搅拌过夜。 然后将反应混合物用更多二氯甲烷稀释，用1N HCl洗涤两次，用盐水洗涤两次，用硫酸钠干燥，然后真空浓缩。 N-（2-苯乙基）氨基甲酸乙酯2d由市售材料通过常规酰化方法（氯甲酸乙酯/ TEA在DCM中）合成（方案1）。 分离化合物2d，收率为96％，无需进行色谱纯化。
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