作为药物合成中间体，用于医药相关研究与开发。
医药领域（作为药物合成中间体）
合成路线 1（1. 合成：4053-45-6）
产率：98%
合成条件：With hydrogenchloride In water at 0 - 20℃; for 8 h;
实验步骤：在0℃下，将14.6g（0.1mol）8-羟基喹啉，16mL 32％HCl水溶液和16mL（0.1mL）37％甲醛水溶液的混合物用氯化氢气体处理6小时。 将溶液在室温下静置2小时，不搅拌。 得到的黄色固体在过滤器上收集，用90％乙醇洗涤并在真空下干燥，得到5-氯甲基-8-羟基喹啉盐酸盐A（19.0g，98％）：1H NMR（250MHz，CDCl3,5）5.32（s， 2H），7.53（m，1H），7.85（m，2H），8.12（m，1H），9.12（m，1H），9.28（m，1H）。
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