化学合成。
医药
合成路线 1(1. 合成:6967-12-0)
产率:94%
合成条件:With hydrogen In methanol
实验步骤:将6-硝基-1H-吲唑(25g,0.153mmol,市售)和10%Pd / C(2.0g)在MeOH中的混合物在H 2(1atm)下搅拌过夜。 过滤后,浓缩滤液,得到1H-吲唑-6-基胺(18.5g,收率94%),为黄色固体。
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